Design, Synthesis, and Antiviral activity of 1,2,3,4-Tetrahydropyrimidine derivatives acting as novel entry inhibitors to target at “Phe43 cavity” of HIV-1 gp120
Jagadeesh Senapathi, Akhila Bommakanti, Veena Kusuma, Srinivas Vangara, Anand K. Kondapi
Topics & Concepts
ChemistryGlycoproteinPyrimidineStereochemistryHuman immunodeficiency virus (HIV)Viral entrySmall moleculeMoleculeVirusBiophysicsBiochemistryCombinatorial chemistryVirologyViral replicationBiologyOrganic chemistryHIV Research and TreatmentHIV/AIDS drug development and treatmentMonoclonal and Polyclonal Antibodies Research