Novel donepezil-chalcone-rivastigmine hybrids as potential multifunctional anti-Alzheimer's agents: Design, synthesis, in vitro biological evaluation, in vivo and in silico studies
Zhipei Sang, Ping Bai, Yujuan Ban, Keren Wang, Anguo Wu, Jing Mi, Jiaqi Hu, Rui Xu, Gaofeng Zhu, Jianta Wang, Jiquan Zhang, Changning Wang, Zhenghuai Tan, Lei Tang
Topics & Concepts
DonepezilIn vivoPharmacologyChemistryRivastigmineNeuroprotectionIn vitroChalconeBiochemistryDementiaMedicineStereochemistryInternal medicineBiologyDiseaseBiotechnologyCholinesterase and Neurodegenerative DiseasesAlzheimer's disease research and treatmentsComputational Drug Discovery Methods