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An Enantioselective Suzuki–Miyaura Coupling To Form Axially Chiral Biphenols

Robert Pearce-Higgins, Larissa N. Hogenhout, Philip J. Docherty, David M. Whalley, Padon Chuentragool, Najung Lee, Nelson Y. S. Lam, Thomas M. McGuire, Damien Valette, Robert J. Phipps

2022Journal of the American Chemical Society73 citationsDOIOpen Access PDF

Abstract

via diastereomeric salt recrystallization.

Topics & Concepts

ChemistryEnantiopure drugEnantioselective synthesisAxial chiralityChirality (physics)Ligand (biochemistry)Combinatorial chemistrySuzuki reactionOrganic chemistryCatalysisPalladiumReceptorNambu–Jona-Lasinio modelQuarkQuantum mechanicsPhysicsChiral symmetry breakingBiochemistryAxial and Atropisomeric Chirality SynthesisMolecular spectroscopy and chiralityChemical synthesis and alkaloids
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