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Guided multi-objective generative AI to enhance structure-based drug design

Amit Kadan, Kevin Ryczko, Erika Lloyd, Adrián E. Roitberg, Takeshi Yamazaki

2025Chemical Science12 citationsDOIOpen Access PDF

Abstract

IDOLpro is a modular framework for guided diffusion which can generate molecules with a plurality of optimized properties for structure-based drug design, accelerating the drug discovery process.

Topics & Concepts

Generative grammarDrugComputer scienceGenerative DesignArtificial intelligenceMedicinePharmacologyEngineeringChemical engineeringCompatibility (geochemistry)Computational Drug Discovery MethodsMachine Learning in Materials ScienceProcess Optimization and Integration
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