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Design and characterization of PROTAC degraders specific to protein N-terminal methyltransferase 1

Qilong Zhou, Wei Wu, Kaimin Jia, Guangyan Qi, Xiuzhi Susan Sun, Ping Li

2022European Journal of Medicinal Chemistry17 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryCell growthCancer researchCalreticulinFusion proteinMethyltransferaseCell cultureMethylationEpigeneticsCell biologyBiochemistryBiologyGeneticsRecombinant DNAGeneEndoplasmic reticulumProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisCancer-related gene regulation
Design and characterization of PROTAC degraders specific to protein N-terminal methyltransferase 1 | Litcius