Design, synthesis and bioactivity evaluation of thiazolidinedione derivatives as partial agonists targeting PPARγ
Juan Sun, Hanyu Liu, Yiheng Zhang, Ze-Yu Fang, Peng‐Cheng Lv
Topics & Concepts
ChemistryThiazolidinedioneAgonistPeroxisome proliferator-activated receptorPartial agonistPharmacologyDocking (animal)PioglitazoneReceptorBiochemistryEndocrinologyBiologyDiabetes mellitusMedicineType 2 diabetesNursingPeroxisome Proliferator-Activated ReceptorsEicosanoids and Hypertension PharmacologyReceptor Mechanisms and Signaling