Identification of a new class of potent aldose reductase inhibitors: Design, microwave-assisted synthesis, in vitro and in silico evaluation of 2-pyrazolines
Belgin Sever, Mehlika Dilek Altıntop, Yeliz Demir, Nalan Yılmaz, Gülşen Akalın Çiftçi, Şükrü Beydemir, Ahmet Özdemır
Topics & Concepts
Aldose reductaseIC50ChemistryAldose reductase inhibitorIn silicoCytotoxicityMoietyPharmacologyBioavailabilityIn vitroDocking (animal)StereochemistrySorbinilPyrazolineBiochemistryEnzymeMedicineMedicinal chemistryGeneNursingAldose Reductase and TaurineEnzyme function and inhibitionSynthesis and Characterization of Pyrroles