Enzyme kinetics and inhibition parameters of human leukocyte glucosylceramidase
Mesut Karataş, Şenol Doğan, Emrulla Spahiu, Adna Ašić, Larisa Bešić, Yusuf Turan
Abstract
of 55.3 mM. This is the first report for the inhibitory effect of glucose, δ-gluconolactone on human leukocyte GCase activity.
Topics & Concepts
EnzymeGlucocerebrosideIC50CeramideEnzyme kineticsBiochemistryChemistryGlucocerebrosidaseUncompetitive inhibitorEnzyme assayActive siteNon-competitive inhibitionIn vitroApoptosisLysosomal Storage Disorders ResearchCarbohydrate Chemistry and SynthesisTrypanosoma species research and implications