Litcius/Paper detail

Design, synthesis and biological evaluation of novel deoxyvasicinone-indole as multi-target agents for Alzheimer’s disease

Ashok Nerella, Madhukar Jeripothula

2021Bioorganic & Medicinal Chemistry Letters27 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryButyrylcholinesteraseAcetylcholinesteraseIndole testPharmacophoreAchéIC50Lead compoundStereochemistryDocking (animal)PharmacologyEnzymeCombinatorial chemistryBiochemistryIn vitroNursingMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity