Synthesis, biological screening and computational analysis of Thiazole linked Thiazolidinone Schiff bases as anti-Alzheimer's drug candidates
Thoraya A. Farghaly, Wajid Rehman, Yousaf Khan, Hina Sarfraz
Topics & Concepts
ChemistryButyrylcholinesteraseAcetylcholinesteraseThiazoleDocking (animal)StereochemistryIC50HOMO/LUMOSchiff baseDonepezilAchéEnzymeCombinatorial chemistryBiochemistryIn vitroOrganic chemistryMoleculeMedicineDiseasePathologyDementiaNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsSynthesis and biological activity