Design, synthesis and biological evaluation of novel quinazoline-derived EGFR/HER-2 dual-target inhibitors bearing a heterocyclic-containing tail as potential anti-tumor agents
Shuang Hao, Jiahui Wang, Liang Hou, Jingwei Liang, Jing-han Yan, Yi-fan Niu, Xinyang Li, Qi Sun, Fan‐hao Meng
Topics & Concepts
QuinazolineChemistryIn vitroEGFR inhibitorsEpidermal growth factor receptorDual (grammatical number)IsozymeInhibitory postsynaptic potentialCombinatorial chemistryStereochemistryBiochemistryEnzymeReceptorNeuroscienceBiologyLiteratureArtHER2/EGFR in Cancer ResearchCancer therapeutics and mechanismsQuinazolinone synthesis and applications