Design and synthesis of new 1,4,5-trisubstituted triazole-bearing benzenesulphonamide moiety as selective COX-2 inhibitors
Mohamed S. Bekheit, Hanan A. Mohamed, Bakr F. Abdel‐Wahab, Marwa A. Fouad
Topics & Concepts
ChemistryPharmacophoreMoietyStereochemistrySelectivityTriazole1,2,3-TriazoleIn silicoIn vitroHydrazideCombinatorial chemistryBiochemistryOrganic chemistryCatalysisGeneSynthesis and biological activityClick Chemistry and ApplicationsInflammatory mediators and NSAID effects