Design, synthesis and in silico insights of novel 1,2,3-triazole benzenesulfonamide derivatives as potential carbonic anhydrase IX and XII inhibitors with promising anticancer activity
Marwa M. Abdelhakeem, Martha M. Morcoss, Dina Hanna, Phoebe F. Lamie
Topics & Concepts
ChemistryADMECarbonic anhydraseLipinski's rule of fiveAcetazolamideCell cultureDocking (animal)StereochemistryIn silicoIC50In vitroEnzymeBiochemistryBiologyGeneMedicineNursingGeneticsAnesthesiaEnzyme function and inhibitionSynthesis and Catalytic ReactionsPhenothiazines and Benzothiazines Synthesis and Activities