Litcius/Paper detail

How can we improve the design of small molecules to target thioredoxin reductase for treating cancer?

Jianqiang Xu, Jianguo Fang

2020Expert Opinion on Drug Discovery20 citationsDOIOpen Access PDF

Abstract

The ubiquitous thioredoxin reductase (TrxR, encoded by TXNRD gene) enzymes are essential to maintain the cellular redox homeostasis. The most outstanding function of TrxR is to keep its native subs...

Topics & Concepts

Thioredoxin reductaseThioredoxinFunction (biology)ReductaseBiologyComputational biologyEnzymeGeneCell biologyBiochemistryRedox biology and oxidative stressMetal-Catalyzed Oxygenation MechanismsEnzyme function and inhibition