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Palladium(<scp>ii</scp>)-catalyzed intramolecular C–H amination to carbazole: the crucial role of cyclic diacyl peroxides

Ting Yuan, Kang Fu, Lei Shi

2024Organic Chemistry Frontiers12 citationsDOI

Abstract

Herein, we have developed an efficient Pd II -catalyzed intramolecular oxidative C–H amination under additive-free and green conditions where strained cyclic diacyl peroxide functions as both a sacrificial oxidant and a bidentate linker.

Topics & Concepts

ChemistryIntramolecular forceAminationPalladiumCatalysisCarbazoleLinkerOxidative phosphorylationDenticityPeroxideCombinatorial chemistryMedicinal chemistryOrganic chemistryMetalBiochemistryComputer scienceOperating systemCatalytic C–H Functionalization MethodsSynthesis and Catalytic ReactionsSulfur-Based Synthesis Techniques
Palladium(<scp>ii</scp>)-catalyzed intramolecular C–H amination to carbazole: the crucial role of cyclic diacyl peroxides | Litcius