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Design, Synthesis, and Anticancer Potential of the Enzyme (PARP-1) Inhibitor with Computational Studies of New Triazole, Thiazolidinone, - Thieno [2, 3-d] Pyrimidinones

Ameen A. Abu‐Hashem, Khadiga M. Abu‐Zied, Magdi E. A. Zaki, Mohamed F. El Shehry, Hanem M. Awad, Mohammed A. Khedr

2020Letters in Drug Design & Discovery30 citationsDOI

Topics & Concepts

ChemistryPyrimidinonesCombinatorial chemistryDPPHAntioxidantStereochemistryQuantitative structure–activity relationshipDocking (animal)Organic chemistryNursingMedicinePARP inhibition in cancer therapyCancer therapeutics and mechanismsSynthesis and biological activity
Design, Synthesis, and Anticancer Potential of the Enzyme (PARP-1) Inhibitor with Computational Studies of New Triazole, Thiazolidinone, - Thieno [2, 3-d] Pyrimidinones | Litcius