Azepino-indazoles as calcitonin gene-related peptide (CGRP) receptor antagonists
Stephen E. Mercer, Prasad V. Chaturvedula, Charles M. Conway, Deborah A. Cook, Carl D. Davis, Sokhom S. Pin, Robert Macci, Richard Schartman, Laura J. Signor, Kimberly A. Widmann, Valerie Whiterock, Ping Chen, Cen Xu, John J. Herbst, Walter A. Kostich, George Thalody, John E. Macor, Gene M. Dubowchik
Topics & Concepts
Calcitonin gene-related peptideBioavailabilityChemistryMigrainePharmacologyCalcitoninIn vivoAntagonistReceptorOral administrationPeptideInternal medicineBiochemistryNeuropeptideMedicineBiologyBiotechnologyMigraine and Headache StudiesTrigeminal Neuralgia and TreatmentsNeuroscience of respiration and sleep