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Azeliragon inhibits PAK1 and enhances the therapeutic efficacy of AKT inhibitors in pancreatic cancer

Weikang Kong, Lingxia Zhu, Tian Li, Jiao Chen, Bo Fan, Wenjing Ji, Chunli Zhang, Xueting Cai, Chunping Hu, Xiaoyan Sun, Peng Cao

2023European Journal of Pharmacology10 citationsDOI

Topics & Concepts

Pancreatic cancerPAK1Cancer researchCancerProtein kinase BKinaseIn vivoMedicineCancer cellApoptosisMalignancyInternal medicineBiologyBiochemistryBiotechnologyCancer Mechanisms and TherapyPancreatic and Hepatic Oncology ResearchHistone Deacetylase Inhibitors Research
Azeliragon inhibits PAK1 and enhances the therapeutic efficacy of AKT inhibitors in pancreatic cancer | Litcius