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Design, synthesis and biological evaluation of cinnamamide-quinazoline derivatives as potential EGFR inhibitors to reverse T790M mutation

Bin Zhang, Zichen Xu, Qingqing Liu, Shengjin Xia, Zhikun Liu, Zhi‐Xin Liao, Shaohua Gou

2021Bioorganic Chemistry22 citationsDOI

Topics & Concepts

ChemistryQuinazolineT790MMutantDocking (animal)EGFR inhibitorsProtein kinase BBiochemistryGefitinibEpidermal growth factor receptorApoptosisStereochemistryReceptorNursingMedicineGeneQuinazolinone synthesis and applicationsCancer therapeutics and mechanismsPeptidase Inhibition and Analysis
Design, synthesis and biological evaluation of cinnamamide-quinazoline derivatives as potential EGFR inhibitors to reverse T790M mutation | Litcius