Litcius/Paper detail

Discovery of multifunctional anti-Alzheimer’s agents with a unique mechanism of action including inhibition of the enzyme butyrylcholinesterase and γ-aminobutyric acid transporters

Anna Pasieka, Dawid Panek, Jakub Jończyk, Justyna Godyń, Natalia Szałaj, Gniewomir Latacz, Julia Tabor, Eva Mezeiová, Fabien Chantegreil, José Dias, Damijan Knez, Junfeng Lu, Rongbiao Pi, Jan Korábečný, Xavier Brazzolotto, Stanislav Gobec, Georg Höfner, Klaus T. Wanner, Anna Więckowska, Barbara Malawska

2021European Journal of Medicinal Chemistry24 citationsDOIOpen Access PDF

Topics & Concepts

ButyrylcholinesteraseChemistryMechanism of actionEnzymeTransporterMechanism (biology)BiochemistryEnzyme inhibitionPharmacologyAcetylcholinesteraseIn vitroAchéGeneBiologyPhilosophyEpistemologyCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments