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Chiral Lewis acid catalysis in a visible light-triggered cycloaddition/rearrangement cascade

Simone Stegbauer, Christian Jandl, Thorsten Bach

2022Chemical Science21 citationsDOIOpen Access PDF

Abstract

Chiral Lewis acid catalysis enables the formation of enantioenriched polycyclic benzoisochromenes 2 from simple 1-naphthaldehydes 1 in an efficient cascade process triggered by a visible light-initiated ortho photocycloaddition.

Topics & Concepts

CascadeCascade reactionChemistryCatalysisDominoCycloadditionYield (engineering)MoleculePhotochemistryLewis acids and basesCombinatorial chemistryStereochemistryOrganic chemistryMaterials scienceMetallurgyChromatographyRadical Photochemical ReactionsOxidative Organic Chemistry ReactionsCatalytic C–H Functionalization Methods
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