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Enzymatic activation of pyruvate kinase increases cytosolic oxaloacetate to inhibit the Warburg effect

Elizabeth K. Wiese, Sadae Hitosugi, Sharon T. Loa, Annapoorna Sreedhar, Lindsey G. Andres‐Beck, Kiran Kurmi, Yuan‐Ping Pang, Larry M. Karnitz, Wilson I. Gonsalves, Taro Hitosugi

2021Nature Metabolism57 citationsDOIOpen Access PDF

Topics & Concepts

PKM2Warburg effectLactate dehydrogenase AGlycolysisPyruvate kinaseLactate dehydrogenaseActivator (genetics)Cancer cellBiochemistryCitrate synthaseAnaerobic glycolysisBiologyChemistryEnzymeCancer researchCancerReceptorGeneticsCancer, Hypoxia, and MetabolismMitochondrial Function and PathologyATP Synthase and ATPases Research
Enzymatic activation of pyruvate kinase increases cytosolic oxaloacetate to inhibit the Warburg effect | Litcius