Litcius/Paper detail

UNC5293, a potent, orally available and highly MERTK-selective inhibitor

Hongchao Zheng, Jichen Zhao, Bing Li, Weihe Zhang, Michael A. Stashko, Katherine A. Minson, Madeline G. Huey, Yubai Zhou, H. Shelton Earp, Dmitri Kireev, Douglas K. Graham, Deborah DeRyckere, Stephen V. Frye, Xiaodong Wang

2021European Journal of Medicinal Chemistry17 citationsDOIOpen Access PDF

Topics & Concepts

MERTKChemistryPharmacologyTyrosine-kinase inhibitorTyrosine kinaseCancer researchReceptor tyrosine kinaseReceptorBiochemistryMedicineCancerInternal medicinePhagocytosis and Immune RegulationErythrocyte Function and PathophysiologyCell death mechanisms and regulation