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Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probes

Jingjing Chen, Yalei Li, Jie Zhang, Minmin Zhang, Aihuan Wei, Hong‐Chun Liu, Zhicheng Xie, Wenming Ren, Wenwen Duan, Zhuo Zhang, Aijun Shen, Youhong Hu

2020European Journal of Medicinal Chemistry54 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryPharmacophoreBRD4EpigeneticsBromodomainHDAC1HistoneHDAC6AcetylationHistone deacetylaseCell biologyCancer researchBiochemistryBiologyDNAGeneProtein Degradation and InhibitorsHistone Deacetylase Inhibitors ResearchPeptidase Inhibition and Analysis
Discovery of selective HDAC/BRD4 dual inhibitors as epigenetic probes | Litcius