Metabolic Stability of the Demyelination Positron Emission Tomography Tracer [18F]3-Fluoro-4-Aminopyridine and Identification of Its Metabolites
Yang Sun, Karla M. Ramos‐Torres, Pedro Brugarolas
Topics & Concepts
ChemistryCYP2E1Metabolism4-AminopyridineCytochrome P450In vivoPositron emission tomographyEnzymeMetabolic stabilityDrug metabolismBiochemistryPharmacologyIn vitroBiophysicsMedicineNuclear medicineBiologyBiotechnologyPotassium channelChemical Reactions and IsotopesRadiopharmaceutical Chemistry and ApplicationsPharmacogenetics and Drug Metabolism