Copper-catalyzed asymmetric [4+1] annulation of yne‑allylic esters with pyrazolones
Guang Xu, Cuiju Zhu, Xiang Li, Kexin Zhu, Hao Xu, Hao Xu
Topics & Concepts
PyrazolonesAllylic rearrangementAnnulationCatalysisCopperChemistryOrganic chemistryMedicinal chemistryStereochemistryAxial and Atropisomeric Chirality SynthesisCatalytic C–H Functionalization MethodsCatalytic Alkyne Reactions