Discovery of juglone and its derivatives as potent SARS-CoV-2 main proteinase inhibitors
Jiahua Cui, Jinping Jia
Topics & Concepts
ChemistryVero cellEnzymeJugloneDocking (animal)IC50StereochemistryProteaseBiochemistryViral replicationStructure–activity relationshipEnzyme inhibitorActive siteIn vitroVirusVirologyBiologyNursingMedicineBioactive Compounds and Antitumor AgentsComputational Drug Discovery MethodsCancer therapeutics and mechanisms