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Design, synthesis, and biological evaluation of 6-(imidazo[1,2-a] pyridin-6-yl) quinazolin-4(3H)-one derivatives as potent anticancer agents by dual targeting Aurora kinase and ROR1

Yanhua Fan, Feng Zhang, Xiong Liang, Mingzhi Su, Fang Luo, Mei Li, Qing Li, Ting Zhong, Meitao Yuan, Yongnan Xu, Shu‐Zhen Mu, Huarong Yang

2023Bioorganic Chemistry21 citationsDOI

Topics & Concepts

ChemistryAurora inhibitorKinaseAurora kinaseApoptosisCell growthAurora B kinaseCancer cellCell cycleCancer researchCancerCellBiochemistryBiologyCell divisionInternal medicineMedicineSpindle apparatusMicrotubule and mitosis dynamicsBacteriophages and microbial interactionsProtist diversity and phylogeny
Design, synthesis, and biological evaluation of 6-(imidazo[1,2-a] pyridin-6-yl) quinazolin-4(3H)-one derivatives as potent anticancer agents by dual targeting Aurora kinase and ROR1 | Litcius