Discovery of A031 as effective proteolysis targeting chimera (PROTAC) androgen receptor (AR) degrader for the treatment of prostate cancer
Linrong Chen, Liuquan Han, Shujun Mao, Ping Xu, Xinxin Xu, Ruibo Zhao, Zhihua Wu, Kai Zhong, Guangliang Yu, Xiaolei Wang
Topics & Concepts
Androgen receptorProstate cancerChemistryProteolysisLNCaPReceptorCancer researchZebrafishChimera (genetics)ProstateAndrogenCancerPharmacologyInternal medicineBiochemistryBiologyHormoneEnzymeMedicineGeneProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysMultiple Myeloma Research and Treatments