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Bestatin analogs-4-quinolinone hybrids as antileishmanial hits: Design, repurposing rational, synthesis, in vitro and in silico studies

Ahmed H.E. Hassan, Kazem Mahmoud, Trong-Nhat Phan, Moataz A. Shaldam, Chae Hyeon Lee, Yeon Ju Kim, Soo Bin Cho, Waleed A. Bayoumi, Selwan M. El‐Sayed, Yeonwoo Choi, Suyeon Moon, Joo Hwan No, Yong Sup Lee, Yong Sup Lee

2023European Journal of Medicinal Chemistry19 citationsDOI

Topics & Concepts

In silicoLeishmania donovaniChemistryIn vitroQuinoloneHybridComputational biologyStereochemistryPharmacologyCombinatorial chemistryBiochemistryLeishmaniasisBiologyVisceral leishmaniasisGeneticsGeneBotanyAntibioticsResearch on Leishmaniasis StudiesPeptidase Inhibition and AnalysisSynthesis and Biological Evaluation
Bestatin analogs-4-quinolinone hybrids as antileishmanial hits: Design, repurposing rational, synthesis, in vitro and in silico studies | Litcius