Exploring the cytotoxic effect and CDK-9 inhibition potential of novel sulfaguanidine-based azopyrazolidine-3,5-diones and 3,5-diaminoazopyrazoles
Ebtehal M. Husseiny, Hamada S. Abulkhair, Nehad M. El‐Dydamony, Kurls E. Anwer
Topics & Concepts
ChemistryCytotoxicityCytotoxic T cellCyclin-dependent kinaseIC50StereochemistryDocking (animal)Cancer cellCDK inhibitorCell cycleIn vitroBiochemistryApoptosisCancerBiologyMedicineGeneticsNursingSynthesis and Biological EvaluationClick Chemistry and ApplicationsSynthesis and biological activity