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Allosteric interactions in the parathyroid hormone GPCR–arrestin complex formation

Lisa J. Clark, James Krieger, Alex D. White, Vasyl Bondarenko, Saifei Lei, Fei Fang, Ji Young Lee, Pemra Doruker, Thore Böttke, Frédéric Jean‐Alphonse, Pei Tang, Thomas J. Gardella, Kunhong Xiao, Ieva Sutkevičiu̅tė, Irene Coin, İvet Bahar, Jean‐Pierre Vilardaga

2020Nature Chemical Biology65 citationsDOIOpen Access PDF

Topics & Concepts

ArrestinParathyroid hormone receptorG protein-coupled receptorAllosteric regulationTransmembrane domainParathyroid hormoneChemistryReceptorBiophysicsBiochemistryCell biologyBiologyHormone receptorGeneticsBreast cancerOrganic chemistryCancerCalciumReceptor Mechanisms and SignalingMass Spectrometry Techniques and ApplicationsProtein Kinase Regulation and GTPase Signaling
Allosteric interactions in the parathyroid hormone GPCR–arrestin complex formation | Litcius