Litcius/Paper detail

Recent insight into the biological activities and SAR of quinolone derivatives as multifunctional scaffold

Vishal Sharma, Rina Das, Dinesh Kumar Mehta, Sumeet Gupta, Katharigatta N. Venugopala, Raghu Prasad Mailavaram, Anroop B. Nair, Ashok K. Shakya, Pran Kishore Deb

2022Bioorganic & Medicinal Chemistry51 citationsDOIOpen Access PDF

Topics & Concepts

QuinoloneScaffoldChemistryDrug discoveryStructure–activity relationshipCombinatorial chemistrySmall moleculeComputational biologyPharmacologyIn vitroAntibioticsBiochemistryBiologyMedicineBiomedical engineeringCancer therapeutics and mechanismsSynthesis and Biological EvaluationSynthesis and biological activity