Apremilast-induced increases in acute ethanol intoxication and decreases in ethanol drinking in mice involve PKA phosphorylation of GABAA β3 subunits
Yuri A. Blednov, Adriana Da Costa, Sonia Mason, Jody Mayfield, Stephen J. Moss, Robert O. Messing
Topics & Concepts
AtaxiaPharmacologyApremilastGABAA receptorEthanolChemistryPhosphorylationInverse agonistEndocrinologyMedicineAgonistInternal medicineReceptorBiochemistryPsychiatryPsoriatic arthritisDiseaseNeuroscience and Neuropharmacology ResearchMemory and Neural MechanismsPhosphodiesterase function and regulation