Litcius/Paper detail

Developing novel classes of protein kinase CK1δ inhibitors by fusing [1,2,4]triazole with different bicyclic heteroaromatic systems

Ilenia Grieco, Maicol Bissaro, Davide Benedetto Tiz, Daniel I. Pérez, Conception Perez, Ana Martı́nez, Sara Redenti, Elena Mariotto, Roberta Bortolozzi, Giampietro Viola, Giorgio Cozza, Giampiero Spalluto, Stefano Moro, Stephanie Federico

2021European Journal of Medicinal Chemistry17 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryMoietyBicyclic moleculeStereochemistryKinaseMolecular modelProtein kinase APyrimidineTriazoleBiochemistryOrganic chemistryProtein Kinase Regulation and GTPase SignalingSynthesis and Characterization of Heterocyclic CompoundsSynthesis and Reactivity of Heterocycles