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Single-molecule analysis reveals agonist-specific dimer formation of µ-opioid receptors

Jan Møller, Ali Işbilir, Titiwat Sungkaworn, Brendan Osberg, Christos Karathanasis, Vikram Sunkara, Eugene O. Grushevskyi, Andreas Böck, Paolo Annibale, Mike Heilemann, Christof Schütte, Martin J. Lohse

2020Nature Chemical Biology128 citationsDOI

Topics & Concepts

G protein-coupled receptorDAMGODimerAgonistReceptorChemistryInternalizationBiophysicsSignal transductionCell biologyBiochemistryOpioid receptorBiologyOrganic chemistryReceptor Mechanisms and SignalingMonoclonal and Polyclonal Antibodies ResearchNeuropeptides and Animal Physiology
Single-molecule analysis reveals agonist-specific dimer formation of µ-opioid receptors | Litcius