Consideration of albumin-mediated hepatic uptake for highly protein-bound anionic drugs: Bridging the gap of hepatic uptake clearance between in vitro and in vivo
Seiji Miyauchi, Soojin Kim, Wooin Lee, Yuichi Sugiyama
Topics & Concepts
AlbuminIn vivoChemistryPharmacologyDrug metabolismIn vitroSerum albuminEffluxPlasma protein bindingDrugBiochemistryMetabolismMedicineBiologyBiotechnologyDrug Transport and Resistance MechanismsProtein Interaction Studies and Fluorescence AnalysisAntibiotics Pharmacokinetics and Efficacy