Litcius/Paper detail

Synthesis of Novel Furo[3,2‐c]coumarin Derivatives through Multicomponent [4+1] Cycloaddition Reaction Using ZnO/FAp as a Sustainable Catalyst

Nagaraju Kerru, Lalitha Gummidi, Kranthi Kumar Gangu, Suresh Maddila, Sreekantha B. Jonnalagadda

2020ChemistrySelect35 citationsDOI

Abstract

Abstract An efficient green protocol is developed for the synthesis of ten new furo[3,2‐c]coumarin derivatives employing zinc oxide loaded on fluorapatite (ZnO/FAp) as catalyst. The three‐component one‐pot condensation occurs between the 4‐hydroxycoumarin, isocyanide and selected aldehyde in ethanol solvent at room temperature. Excellent yields (94‐98 %) of target products in 16‐20 min reaction time is the attractive feature. As‐synthesized catalysts and organic compounds were fully established by powder‐XRD, TEM, SEM, EDX, FT‐IR, BET, HRMS, 1 H NMR and 13 C NMR analysis. The catalyst is recyclable up to five times with high efficacy and marginal loss of activity. The reaction facilitated 98 % of the atom economy and 100 % carbon efficiency. Other advantages of the protocol are mild reaction conditions, easy‐workup, green solvent, catalyst reusability, and chromatography free products.

Topics & Concepts

CatalysisAldehydeChemistryCycloadditionCondensation reactionCoumarinSolventAtom economyZincCarbon-13 NMRNuclear chemistryOrganic chemistryMulticomponent Synthesis of HeterocyclesSynthesis and biological activitySynthesis and Biological Evaluation
Synthesis of Novel Furo[3,2‐c]coumarin Derivatives through Multicomponent [4+1] Cycloaddition Reaction Using ZnO/FAp as a Sustainable Catalyst | Litcius