PNU-120596, a positive allosteric modulator of α7 nicotinic acetylcholine receptor, directly inhibits p38 MAPK
Junsuke Uwada, Hitomi Nakazawa, Daisuke Mikami, Mohammad Sayful Islam, Ikunobu Muramatsu, Takanobu Taniguchi, Takashi Yazawa
Topics & Concepts
Methyllycaconitinep38 mitogen-activated protein kinasesMAPK/ERK pathwayPhosphorylationCell biologyChemistryKinaseNicotinic agonistPharmacologyBiologyNicotinic acetylcholine receptorReceptorBiochemistryNicotinic Acetylcholine Receptors StudyComputational Drug Discovery MethodsReceptor Mechanisms and Signaling