Novel quinazoline-based EGFR kinase inhibitors: A review focussing on SAR and molecular docking studies (2015-2019)
Parth Bhatia, Vrinda Sharma, Ozair Alam, Ajay Manaithiya, Perwaiz Alam, Kahksha, Md Tauquir Alam, Mohd Imran
Topics & Concepts
QuinazolineEGFR inhibitorsOsimertinibDocking (animal)Epidermal growth factor receptorDrug discoveryComputational biologyChemistryCancerErlotinibBioinformaticsMedicineBiologyInternal medicineCombinatorial chemistryNursingLung Cancer Treatments and MutationsQuinazolinone synthesis and applicationsCancer therapeutics and mechanisms