In silico identification of noncompetitive inhibitors targeting an uncharacterized allosteric site of falcipain-2
Jorge Enrique Hernández González, Emir Salas‐Sarduy, Lilian Hernández Alvarez, Diego E. B. Gomes, Pedro G. Pascutti, Chris Oostenbrink, Vitor B. P. Leite
Topics & Concepts
Allosteric regulationIn silicoBinding siteVirtual screeningActive siteEnzymeSmall moleculeChemistryNon-competitive inhibitionBiochemistryStereochemistryDrug discoveryGeneRNA and protein synthesis mechanismsTrypanosoma species research and implicationsBiochemical and Structural Characterization