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Structure Based Design of Some Novel 3-Methylquinoxaline Derivatives Through Molecular Docking and Pharmacokinetics Studies as Novel VEGFR-2 Inhibitors

Sagiru Hamza Abdullahi, Adamu Uzairu, Gideon Adamu Shallangwa, Sani Uba, Abdullahi Bello Umar

2022Chemistry Africa15 citationsDOI

Topics & Concepts

Docking (animal)SorafenibDrugChemistryPharmacokineticsPharmacologyStereochemistryProtein Data Bank (RCSB PDB)Lipinski's rule of fiveCombinatorial chemistryComputational biologyMedicineInternal medicineIn silicoBiologyBiochemistryHepatocellular carcinomaGeneNursingSynthesis and Biological EvaluationSynthesis and biological activityQuinazolinone synthesis and applications
Structure Based Design of Some Novel 3-Methylquinoxaline Derivatives Through Molecular Docking and Pharmacokinetics Studies as Novel VEGFR-2 Inhibitors | Litcius