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Biological evaluation of non-basic chalcone CYB-2 as a dual ABCG2/ABCB1 inhibitor

Chao‐Yun Cai, Wei Zhang, Jing‐Quan Wang, Zi‐Ning Lei, Yunkai Zhang, Yi‐Jun Wang, Pranav Gupta, Cai‐Ping Tan, Bo Wang, Zhe‐Sheng Chen

2020Biochemical Pharmacology38 citationsDOI

Topics & Concepts

ChalconeAbcg2EffluxATP-binding cassette transporterMultiple drug resistanceTransporterPharmacologyChemistryBiochemistryBiologyStereochemistryGeneAntibioticsDrug Transport and Resistance MechanismsCancer therapeutics and mechanismsMetal complexes synthesis and properties
Biological evaluation of non-basic chalcone CYB-2 as a dual ABCG2/ABCB1 inhibitor | Litcius