Imatinib can act as an Allosteric Activator of Abl Kinase
Tao Xie, Tamjeed Saleh, P. Rossi, Darcie J. Miller, Charalampos G. Kalodimos
Topics & Concepts
Allosteric regulationImatinibABLChemistryImatinib mesylateActivator (genetics)Chronic myelogenous leukemiaBiologyBiochemistryCancer researchLeukemiaTyrosine kinaseEnzymeReceptorGeneticsMyeloid leukemiaChronic Myeloid Leukemia TreatmentsEosinophilic Disorders and SyndromesQuinazolinone synthesis and applications