Exploring phenylcarbamoylazinane-1,2,4-triazole thioethers as lipoxygenase inhibitors supported with in vitro, in silico and cytotoxic studies
Wardah Shahid, Muhammad Ashraf, Muhammad Saleem, Bushra Bashir, Saima Muzaffar, Mudassar Ali, Ayesha Kaleem, Aziz-ur- Rehman, Hira Amjad, Keshab Bhattarai, Naheed Riaz
Topics & Concepts
ChemistryStereochemistryMTT assayIn silicoIC50HydrazideLipoxygenaseIn vitroCytotoxicityViability assayEnzymeBiochemistryOrganic chemistryGeneSynthesis and Biological EvaluationSynthesis and biological activityClick Chemistry and Applications