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A phase I study of an oral selective gamma secretase (GS) inhibitor RO4929097 in combination with neoadjuvant paclitaxel and carboplatin in triple negative breast cancer

Sagar Sardesai, Mohamed Badawi, Ewa Mrózek, Evan Morgan, Mitch A. Phelps, Julie Stephens, Lai Wei, Mahmoud Kassem, Yonghua Ling, Maryam B. Lustberg, Daniel G. Stover, Nicole Williams, Rachel M. Layman, Raquel E. Reinbolt, Jeffrey VanDeusen, Mathew Cherian, Michael R. Grever, William E. Carson, Bhuvaneswari Ramaswamy, Robert Wesolowski

2020Investigational New Drugs36 citationsDOIOpen Access PDF

Topics & Concepts

MedicineCarboplatinNeutropeniaPaclitaxelInternal medicineBreast cancerGastroenterologyDiscontinuationFebrile neutropeniaPharmacokineticsChemotherapyCmaxCancerOncologyPharmacologyUrologyCisplatinBreast Cancer Treatment StudiesHER2/EGFR in Cancer ResearchCancer Cells and Metastasis
A phase I study of an oral selective gamma secretase (GS) inhibitor RO4929097 in combination with neoadjuvant paclitaxel and carboplatin in triple negative breast cancer | Litcius