Hydrophobic tag-based protein degradation: Development, opportunity and challenge
Qindi He, Xiaofei Zhao, Donglin Wu, Siming Jia, Canlin Liu, Zitian Cheng, Fei Huang, Yadong Chen, Tao Lu, Shuai Lü
Topics & Concepts
ChemistryComputational biologyProtein degradationProteolysisDrug discoverySmall moleculeDegradation (telecommunications)Drug developmentCombinatorial chemistryDrugPharmacologyBiochemistryEnzymeComputer scienceBiologyMedicineTelecommunicationsProtein Degradation and InhibitorsPeptidase Inhibition and AnalysisUbiquitin and proteasome pathways