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Desymmetrization of difluoromethylene groups by C–F bond activation

Trevor W. Butcher, Jonathan Lee Yang, Willi M. Amberg, Nicholas B. Watkins, Natalie D. Wilkinson, John F. Hartwig

2020Nature134 citationsDOIOpen Access PDF

Topics & Concepts

StereocenterEnantioselective synthesisChemistryDesymmetrizationStereochemistryHydrogen bondAllylic rearrangementCatalysisMedicinal chemistryOrganic chemistryMoleculeFluorine in Organic ChemistryAsymmetric Synthesis and CatalysisCyclopropane Reaction Mechanisms
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