Regioselective C5-H direct iodination of indoles
Zhao‐Yang Wang, Rui-Li Guo, Xinglong Zhang, Meng‐Yue Wang, Gang-Ni Chen, Yong‐Qiang Wang
Abstract
An efficient regioselective C5-H direct iodination of indoles is reported herein for the first time, which offers a general and practical access to the difficult C5 functionalization of indoles.
Topics & Concepts
RegioselectivityChemistryHalogenationCombinatorial chemistrySurface modificationOrganic chemistryCatalysisPhysical chemistryCatalytic C–H Functionalization MethodsVanadium and Halogenation ChemistrySynthesis and Catalytic Reactions