Design, synthesis and biological evaluation of novel 2-(4-(1H-indazol-6-yl)-1H-pyrazol-1-yl)acetamide derivatives as potent VEGFR-2 inhibitors
Xingrong Wang, Shuai Wang, Wenbo Li, Kai-Yan Xu, Xue-Peng Qiao, Xue-Li Jing, Zi-Xiao Wang, Changjiang Yang, Shi‐Wu Chen
Topics & Concepts
ChemistryAngiogenesisAcetamideApoptosisCancer researchPI3K/AKT/mTOR pathwayIC50Cancer cellIn vitroMolecular biologyCell biologyStereochemistryBiochemistryCancerBiologyInternal medicineMedicineOrganic chemistryAngiogenesis and VEGF in CancerPI3K/AKT/mTOR signaling in cancerCancer Mechanisms and Therapy